| Company Name: |
TargetMol Chemicals Inc.
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| Tel: |
15002134094 |
| Email: |
marketing@targetmol.cn |
| Products Intro: |
Product Name:M867
CAS:680999-39-7
Package:50mg;5mg
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M867 manufacturers
- M867
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- $0.00 / 50mg
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2025-05-17
- CAS:680999-39-7
- Min. Order:
- Purity:
- Supply Ability: 10g
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| Product Name: | M867 | | Synonyms: | M867;Pentanoic acid, 3-[[(2S)-2-[5-(1,1-dimethylethyl)-3-[[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino]-2-oxo-1(2H)-pyrazinyl]-1-oxobutyl]amino]-5-(methylpentylamino)-4-oxo-, (3S)- | | CAS: | 680999-39-7 | | MF: | C27H43N7O6 | | MW: | 561.67 | | EINECS: | | | Product Categories: | | | Mol File: | 680999-39-7.mol |  |
| density | 1.257±0.14 g/cm3(Temp: 25 °C; Press: 760 Torr)(predicted) | | pka | 3.809±0.19(predicted) |
| Uses | M867 is a selective and reversible inhibitor of caspase-3 with an IC50 of 1.4 nM and Ki of 0.7 nM. M867 has anti apoptotic activity[1]. | | IC 50 | Caspase 3 | | References | [1] Han Y, et.al. Novel pyrazinone mono-amides as potent and reversible caspase-3 inhibitors. Bioorg Med Chem Lett. 2005 Feb 15;15(4):1173-80. DOI:10.1016/j.bmcl.2004.12.006 |
| | M867 Preparation Products And Raw materials |
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